8-Cyclopentyl - 1,3 - dipropylxanthine, solide

Code: c101-25mg D2-231

Non disponible en dehors du Royaume-Uni et de l'Irlande

Application

8-Cyclopentyl-1,3-dipropylxanthine has been used as an adenosine receptor (A1AR) antagonist in macrophages and human umbilical vein endothelial cells (HUVECs). It...


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Votre prix
$105.68 25MG

Non disponible en dehors du Royaume-Uni et de l'Irlande

Application

8-Cyclopentyl-1,3-dipropylxanthine has been used as an adenosine receptor (A1AR) antagonist in macrophages and human umbilical vein endothelial cells (HUVECs). It has also been used as A1AR antagonist in MCF-7 breast cancer cell line to test its anti-cancer effect.

Biochem/physiol Actions

8-Cyclopentyl-1,3-dipropylxanthine (DPCPX) is a selective A1adenosine receptor antagonist. DPCPX possesses anti-cancer functionality. It induces apoptosis in breast cancer cells and favors mRNA expression of caspases.

Features and Benefits

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Packaging

25, 100 mg in poly bottle

εmax14,800 at 276 nm in ethanol
colorwhite
formsolid
Gene Informationhuman ... ADORA1(134), ADORA2A(135), ADORA2B(136), ADORA3(140)rat ... Adora1(29290), Adora2a(25369), Adora2b(29316), Adora3(25370)
InChI keyFFBDFADSZUINTG-UHFFFAOYSA-N
InChI1S/C16H24N4O2/c1-3-9-19-14-12(15(21)20(10-4-2)16(19)22)17-13(18-14)11-7-5-6-8-11/h11H,3-10H2,1-2H3,(H,17,18)
Quality Level100
SMILES stringCCCN1C(=O)N(CCC)c2nc([nH]c2C1=O)C3CCCC3
solubilityethanol: 4 mg/mL, DMSO: >10 mg/mL, H2O: insoluble, 0.1 M NaOH: 2 mg/mL
Code
Description
Unité de vente
Prix annoncé
Qté
C101-100MG
Unité:100MG
Prix annoncé: $316.74
Source:Prix annoncé
Cas Number102146-07-6
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