BQ-788, >=95%, solid

Code: b157-200ug D2-231

Not available outside of the UK & Ireland.

Application

BQ-788 has been used as a selective endothelin-B (ETRB) blocker in human airway smooth muscle cells (HASMCs), uterine mesothelial cells (UtMCs)-derived vascular s...


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£185.00 200UG
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Not available outside of the UK & Ireland.

Application

BQ-788 has been used as a selective endothelin-B (ETRB) blocker in human airway smooth muscle cells (HASMCs), uterine mesothelial cells (UtMCs)-derived vascular smooth muscle cells (VSMCs), and human umbilical vein endothelial cells (HUVECs)

Biochem/physiol Actions

Selective ETB endothelin receptor antagonist.

assay≥95%
colorwhite
formsolid
Gene Informationhuman ... EDNRB(1910)mouse ... EDNRB(13618)rat ... EDNRB(50672)
InChI keyQCVIFBRTTLMEOV-FUKQNADPSA-M
InChI1S/C34H51N5O7.Na/c1-8-9-16-25(31(42)43)35-29(40)26(18-23-20-38(33(45)46-7)28-17-11-10-15-24(23)28)36-30(41)27(19-34(4,5)6)37-32(44)39-21(2)13-12-14-22(39)3;/h10-11,15,17,20-22,25-27H,8-9,12-14,16,18-19H2,1-7H3,(H,35,40)(H,36,41)(H,37,44)(H,42,43);/q;+1/p-1/t21-,22+,25-,26-,27+;/m1./s1
Quality Level200
SMILES string[Na+].CCCC[C@@H](NC(=O)[C@@H](Cc1cn(C(=O)OC)c2ccccc12)NC(=O)[C@H](CC(C)(C)C)NC(=O)N3[C@@H](C)CCC[C@H]3C)C([O-])=O
solubilityDMSO: 1.2 mg/mL, ethanol: 1.2 mg/mL, acetonitrile: 0.3 mg/mL, H2O: slightly soluble
storage temp.−20°C
Cas Number156161-89-6
This product has met the following criteria: